CI 988 (PD134308) 是一种有效的、选择性的、具有口服活性的 CCK2R（胆囊收缩素 2 受体）拮抗剂，对小鼠皮质 CCK2 的 IC50 为 1.7 nM。
| Cas No. | 130332-27-3 |
| 别名 | PD134308 |
| 化学名 | 4-(((R)-2-((R)-2-((((1R,2R,3R,5S,7S)-adamantan-2-yloxy)carbonyl)amino)-3-(1H-indol-3-yl)-2-methylpropanamido)-1-phenylethyl)amino)-4-oxobutanoic acid |
| Canonical SMILES | O=C(N[C@@](C)(C(NC[C@@H](C1=CC=CC=C1)NC(CCC(O)=O)=O)=O)CC2=CNC3=CC=CC=C23)O[C@@H]4[C@H]5C[C@H]6C[C@H]4C[C@H](C6)C5 |
| 分子式 | C35H42N4O6 |
| 分子量 | 614.73 |
| 溶解度 | <61.47mg/ml in DMSO |
| 储存条件 | Store at -20℃ |
| General tips | For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while. |
| Shipping Condition | Evaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request |
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