JTP-117968, a novel selectiveglucocorticoid receptormodulator (a non-steroidal SGRM,IC₅₀of 6.8 nM), exhibits improved transrepression/transactivation dissociation^[1].

JTP-117968 has partial TR activity, but exhibits extremely low TA activity^[1].

520.59

C₃₁H₃₁F₃N₂O₂

2250132-99-9

Room temperature in continental US; may vary elsewhere.

Please store the product under the recommended conditions in the Certificate of Analysis.