SCH 221510 是一种有效的、具有口服活性的选择性 NOP(伤害感受素阿片受体)激动剂,EC50 为 12 nM,Ki 为 0.3 nM。
Cas No. | 322473-89-2 |
化学名 | (1R,3s,5S)-8-(di-o-tolylmethyl)-3-phenyl-8-azabicyclo[3.2.1]octan-3-ol |
Canonical SMILES | O[C@@]1(C2=CC=CC=C2)C[C@H](CC3)N(C(C4=CC=CC=C4C)C5=CC=CC=C5C)[C@H]3C1 |
分子式 | C28H31NO |
分子量 | 397.55 |
溶解度 | <39.76mg/ml in DMSO |
储存条件 | Store at RT |
General tips | For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while. |
Shipping Condition | Evaluation sample solution : ship with blue ice All other available size: ship with RT , or blue ice upon request |
产品描述 | Potent and selective NOP agonist |