CAS NO: | 159768-75-9 |
包装 | 价格(元) |
100mg | 电议 |
250mg | 电议 |
500mg | 电议 |
生物活性 | Lobradimil (RMP 7), a synthetic bradykinin analog, is a potent and selectivebradykinin B2 receptoragonist (Ki: 0.54 nM). Lobradimil increases the permeability of the BBB. Lobradimil can be used in the research of brain tumors[1]. | ||||||||
IC50& Target[1] |
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体外研究 (In Vitro) | Lobradimil induces an increase in intracellular free calcium levels in RBME cells[3]. | ||||||||
体内研究 (In Vivo) | Lobradimil (2.5-mg/kg bolus plus 10 mg/kg/h for 90 minutes) increases brain tumor permeability and shows hypotensive effects in RG2 glioma cells-implanted rats[2].
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Clinical Trial | |||||||||
分子量 | 1098.28 | ||||||||
Formula | C49H75N15O12S | ||||||||
CAS 号 | 159768-75-9 | ||||||||
运输条件 | Room temperature in continental US; may vary elsewhere. | ||||||||
储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |