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(R)-Praziquantel-d11
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
(R)-Praziquantel-d11图片
CAS NO:1399880-38-6
包装与价格:
包装价格(元)
1mg电议
5mg电议
10mg电议
50mg电议
100mg电议

产品名称
(R)-吡喹酮 D11
产品介绍
(R)-Praziquantel D11 是 (R)-Praziquantel 的氘代物。(R)-Praziquantel 是 Praziquantel 的活性对映体,是一种人5-HT2B受体的部分激动剂。(R)-Praziquantel 用作驱虫药,抗血吸虫。
生物活性

(R)-Praziquantel D11 is the deuterium labeled (R)-Praziquantel. (R)-Praziquantel, the active enantiomer of Praziquantel, is a partial agonist of the human 5-HT2B receptor. (R)-Praziquantel acts as an antischistosomal eutomer[1].

IC50& Target[1]

5-HT2BReceptor

 

Antischistosomal

 

体外研究
(In Vitro)

(R)-Praziquantel ((R)-PZQ) is a G-protein-coupled receptor ligand. (R)-Praziquantel modulation of serotoninergic signaling occurs over a concentration range sufficient to regulate vascular tone of the mesenteric blood vessels where the adult parasites reside within their host. The important anthelmintic is supported by a broad, cross species polypharmacology with (R)-Praziquantel modulating signaling events in both host and parasite[1].

分子量

323.47

Formula

C19H13D11N2O2

CAS 号

1399880-38-6

中文名称

(R)-吡喹酮 D11

运输条件

Room temperature in continental US; may vary elsewhere.

储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.