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Risperidone-d4
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
Risperidone-d4图片
CAS NO:1020719-76-9
包装与价格:
包装价格(元)
2.5mg电议
5mg电议

产品名称
R 64 766-d4
产品介绍
Risperidone-d4 (R 64 766-d4) 是 Risperidone 的氘代物。Risperidone是5-HT2受体的阻断剂,P-糖蛋白(P-Glycoprotein)的抑制剂 和dopamine D2受体的拮抗剂,其对 5-HT2A和 dopamine D2受体的Ki值分别为 4.8,5.9 nM。
生物活性

Risperidone-d4 (R 64 766-d4) is the deuterium labeled Risperidone. Risperidone is a serotonin5-HT2receptorblocker,P-Glycoproteininhibitor and potentdopamineD2receptorantagonist, withKisof 4.8, 5.9 nM for 5-HT2Aand dopamineD2receptor, respectively.

体外研究
(In Vitro)

Stable heavy isotopes of hydrogen, carbon, and other elements have been incorporated into drug molecules, largely as tracers for quantitation during the drug development process. Deuteration has gained attention because of its potential to affect the pharmacokinetic and metabolic profiles of drugs[1].

分子量

414.51

性状

Solid

Formula

C23H23D4FN4O2

CAS 号

1020719-76-9

运输条件

Room temperature in continental US; may vary elsewhere.

储存方式
Powder-20°C3 years
In solvent-80°C6 months
-20°C1 month