HDAC6/8/BRPF1-IN-1 is a dual inhibitor of bothHDAC6/8 and the bromodomain and PHD finger containing protein 1 (BRPF1). HDAC6/8/BRPF1-IN-1 has inhibitory activity forHDAC1,HDAC6andHDAC8withIC₅₀values of 797 nM, 344 nM and 908 nM, respectively. HDAC6/8/BRPF1-IN-1 has inhibitory activity forBRPF1with anK_dvalue of 175.2 nM. HDAC6/8/BRPF1-IN-1 can be used for the research ofcancer^[1].

HDAC6/8/BRPF1-IN-1 has inhibitory activity for HDAC1, HDAC6 and HDAC8 with IC₅₀values of 797 nM, 344 nM and 908 nM, respectively^[1].
HDAC6/8/BRPF1-IN-1 has inhibitory activity for BRPF1 with an K_dvalue of 175.2 nM^[1].

387.41

C₁₈H₁₇N₃O₅S

2484255-65-2

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