CDK4/6-IN-12

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CDK4/6-IN-12

本产品不向个人销售，仅用作科学研究，不用于任何人体实验及非科研性质的动物实验。

CAS NO:

2445205-24-1

包装与价格：

包装	价格(元)
100mg	电议
250mg	电议
500mg	电议

产品介绍

CDK4/6-IN-12 是一种有效的周期蛋白依赖性激酶 4/6 抑制剂。CDK4/6-IN-12 对 CDK4 和 CDK6 具有酶抑制活性，IC₅₀值分别为 592.3 nM 和 3090 nM。 CDK4/6-IN-12 可用于癌症的研究。

生物活性

CDK4/6-IN-12 is a potentcyclin-dependent kinase4/6 (CDK4/6)inhibitor. CDK4/6-IN-12 has enzymatic inhibitory activity forCDK4andCDK6withIC₅₀of 592.3 nM and 3090 nM, respectively. CDK4/6-IN-12 can be used for the research ofcancer^[1].

IC₅₀& Target^[1]

CDK4

592.3 nM (IC₅₀)

CDK6

3090 nM (IC₅₀)

体外研究
(In Vitro)

CDK4/6-IN-12 (compound 4a) inhibits CDK4 and CDK6 with IC₅₀of 592.3 nM and 3090 nM, respectively^[1].

分子量

238.25

Formula

C₁₂H₁₀N₆

CAS 号

2445205-24-1

运输条件

Room temperature in continental US; may vary elsewhere.

储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.