SB 243213 dihydrochloride 是一种具有口服活性、选择性和高亲和力的 5-HT2C 受体拮抗剂,对人 5-HT2C 受体的 pKi 为 9.37,pKb 为 9.8。
Cas No. | 200940-23-4 |
化学名 | (Z)-5-methyl-N-(6-((2-methylpyridin-3-yl)oxy)pyridin-3-yl)-6-(trifluoromethyl)indoline-1-carbimidic acid dihydrochloride |
Canonical SMILES | CC1=CC(CCN2/C(O)=N/C3=CN=C(OC(C=CC=N4)=C4C)C=C3)=C2C=C1C(F)(F)F.Cl.Cl |
分子式 | C22H19F3N4O2.2HCl |
分子量 | 501.33 |
溶解度 | <25.07mg/ml in DMSO |
储存条件 | Store at -20℃ |
General tips | For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while. |
Shipping Condition | Evaluation sample solution : ship with blue ice All other available size: ship with RT , or blue ice upon request |