TC LPA5 4 是一种 LPA5 (GPR92) 特异性非脂质拮抗剂。 TC LPA5 4 抑制 LPA 诱导的分离的人血小板（LPA5-RH7777 细胞系）的聚集，IC50 为 800 nM。 TC LPA5 4 显示对 LPA5 超过 80 种其他筛选药物靶点的选择性。 TC LPA5 4 抑制甲状腺癌细胞的细胞增殖和迁移。
| Cas No. | 1393814-38-4 |
| 化学名 | 5-(3-chloro-4-cyclohexylphenyl)-1-(3-methoxyphenyl)-1H-pyrazole-3-carboxylic acid |
| Canonical SMILES | COC1=CC=CC(N2C(C3=CC(Cl)=C(C4CCCCC4)C=C3)=CC(C(O)=O)=N2)=C1 |
| 分子式 | C23H23ClN2O3 |
| 分子量 | 410.89 |
| 溶解度 | <41.09mg/ml in DMSO |
| 储存条件 | Store at -20℃ |
| General tips | For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while. |
| Shipping Condition | Evaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request |
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