| CAS NO: | 1623002-61-8 |
| 包装 | 价格(元) |
| 1mg | 电议 |
| 5mg | 电议 |
| 10mg | 电议 |
| 生物活性 | NTRC-824 (Compound 5) is a potent, selective and neurotensin-like nonpeptideneurotensin receptortype 2 (NTS2)antagonist with anIC50of 38 nM and aKiof 202 nM. NTRC-824 is >150-fold selectivity forNTS2over NTS1 (Ki>30 μM)[1]. | |||||||||
| IC50& Target | IC50: 38 nM (Nurotensin receptor type 2)[1] | |||||||||
| 体外研究 (In Vitro) | Testing of NTRC-824 (Compound 5) at the NTS1 receptor shows no binding activity in the NTS1 assay up to 30 μM, making NTRC-824 (Compound 5) selective for NTS2 in both the binding and functional assays. NTRC-824 (Compound 5) is the first nonpeptide compound that behaves like, and is more active than, the endogenous ligand[1]. | |||||||||
| 分子量 | 553.55 | |||||||||
| 性状 | Solid | |||||||||
| Formula | C25H26F3N3O6S | |||||||||
| CAS 号 | 1623002-61-8 | |||||||||
| 运输条件 | Room temperature in continental US; may vary elsewhere. | |||||||||
| 储存方式 |
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