MCHR1antagonist 3 is a potent themelanin-concentrating hormone receptor-1 (MCHR1)antagonist.MCHR1antagonist 3 is used to regulate energy metabolism^[1].

Compound 1, derived from a spirohydantoin scaffold, exhibits a K_iof 50 nM at MCH-R1. Compound 1 is a potent inhibitor of CYP3A4 (IC₅₀=35 nM). MCHR1 antagonist 3 is an analog of compound 1^[1].

472.62

C₂₉H₃₆N₄O₂

1069622-60-1

Room temperature in continental US; may vary elsewhere.

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