CAS NO: | 92933-48-7 |
包装 | 价格(元) |
100mg | 电议 |
250mg | 电议 |
500mg | 电议 |
生物活性 | LUF6283 is a potent and orally activeHCA(2)partial agonist, with aKiof 0.55 μM. LUF6283 can achieve the beneficial lipid lowering effect of niacin without producing the unwanted cutaneous flushing side effect[1]. |
IC50& Target | EC50: 0.32 ± 0.06 μM (pERK1/2)[1] |
体内研究 (In Vivo) | LUF6283 (C57BL/6 mice, 400 mg/kg, Oral gavage, once a day for 4 weeks) has no effect on adipose tissue ATGL/HSL expression, and significantly reduces the expression of apolipoprotein B (APOB)[1]. |
分子量 | 168.19 |
Formula | C8H12N2O2 |
CAS 号 | 92933-48-7 |
运输条件 | Room temperature in continental US; may vary elsewhere. |
储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |