TPMPA 是 isoguvacine 和 3-APMPA 的混合物,是第一个 GABAC 受体 (KB = 2.1 μM) 的选择性拮抗剂,但不与 GABAA (KB = 320 μM) 或 GABAB 受体 (EC50 = 500 μM) 相互作用。
Cas No. | 182485-36-5 |
化学名 | (R)-methyl(1,2,3,6-tetrahydropyridin-4-yl)phosphinic acid |
Canonical SMILES | O[P@@](C1=CCNCC1)(C)=O |
分子式 | C6H12NO2P |
分子量 | 161.14 |
溶解度 | PBS (pH 7.2): 10 mg/ml |
储存条件 | Store at -20°C |
General tips | For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while. |
Shipping Condition | Evaluation sample solution : ship with blue ice All other available size: ship with RT , or blue ice upon request |