GYKI 52466 dihydrochloride 是一种具有口服活性、高选择性和非竞争性的 AMPA/红藻氨酸受体拮抗剂,IC50 值分别为 7.5 和 11μM。
Cas No. | 102771-26-6 |
别名 | 1-(4-氨基苯基)-4-甲基-7,8亚甲基二氧-5H-2,3-苯并二氮杂卓盐酸盐 |
化学名 | 4-(8-methyl-9H-[1,3]dioxolo[4',5':4,5]benzo[1,2-d][1,2]diazepin-5-yl)aniline |
Canonical SMILES | CC(CC1=CC(OCO2)=C2C=C13)=NN=C3C4=CC=C(N)C=C4 |
分子式 | C17H15N3O2.2HCl |
分子量 | 366.24 |
溶解度 | <16.49mg/ml in DMSO |
储存条件 | Desiccate at RT |
General tips | For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while. |
Shipping Condition | Evaluation sample solution : ship with blue ice All other available size: ship with RT , or blue ice upon request |