Methysticin 是一种从卡瓦根中分离出来的卡瓦内酯。
| Cas No. | 495-85-2 |
| 别名 | 麻醉椒苦素 |
| Canonical SMILES | COC(C[C@H](/C=C/C1=CC=C(OCO2)C2=C1)O3)=CC3=O |
| 分子式 | C15H14O5 |
| 分子量 | 274.3 |
| 溶解度 | DMF: 2.5 mg/mL,DMSO: 5 mg/mL,DMSO:PBS (pH 7.2) (1:6): 0.14 mg/mL,Ethanol: 1 mg/mL |
| 储存条件 | 4°C, protect from light |
| General tips | For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while. |
| Shipping Condition | Evaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request |
| 产品描述 | Methysticin is a natural kavalactone from the kava plant, P. methysticum. It enhances the binding of bicuculline methochloride at the γ-aminobutyric acid (GABA) receptor GABAA at 0.1 µM. Methysticin inhibits the cytochrome P450 (CYP) isoforms CYP2C9 and CYP2D6. |
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