CAS NO: | 23827-91-0 |
包装 | 价格(元) |
5mg | 电议 |
10mg | 电议 |
25mg | 电议 |
50mg | 电议 |
100mg | 电议 |
生物活性 | [Des-Arg9]-Bradykinin acetate is aBradykinin B1receptoragonist that displays selectivity for B1over B2receptors. | ||||||||||||||||
IC50& Target | Bradykinin B1receptor[1] | ||||||||||||||||
体外研究 (In Vitro) | [Des-Arg9]-Bradykinin acetate is a Bradykinin(B1) receptor agonist. The B2receptor mediates the action of bradykinin (BK) and lysyl-bradykinin (Lys-BK), the first set of bioactive kinins formed in response to injury from kininogen precursors through the actions of plasma and tissue kallikreins, whereas the B1receptor mediates the action of [Des-Arg9]-Bradykinin (des-Arg9-BK) and Lys-des-Arg Arg9-BK, the second set of bioactive kinins formed through the actions of carboxypeptidases on BK and Lys-BK, respectively[1]. | ||||||||||||||||
分子量 | 964.07 | ||||||||||||||||
性状 | Solid | ||||||||||||||||
Formula | C46H65N11O12 | ||||||||||||||||
CAS 号 | 23827-91-0 | ||||||||||||||||
Sequence | Arg-Pro-Pro-Gly-Phe-Ser-Pro-Phe | ||||||||||||||||
Sequence Shortening | RPPGFSPF | ||||||||||||||||
中文名称 | [Des-Arg9]-缓激肽醋酸盐 | ||||||||||||||||
运输条件 | Room temperature in continental US; may vary elsewhere. | ||||||||||||||||
储存方式 | Sealed storage, away from moisture
*In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture) | ||||||||||||||||
溶解性数据 | In Vitro: H2O : 100 mg/mL(103.73 mM;Need ultrasonic) 配制储备液
* 请根据产品在不同溶剂中的溶解度选择合适的溶剂配制储备液;一旦配成溶液,请分装保存,避免反复冻融造成的产品失效。 In Vivo: 请根据您的实验动物和给药方式选择适当的溶解方案。以下溶解方案都请先按照In Vitro方式配制澄清的储备液,再依次添加助溶剂: ——为保证实验结果的可靠性,澄清的储备液可以根据储存条件,适当保存;体内实验的工作液,建议您现用现配,当天使用;
以下溶剂前显示的百
*以上所有助溶剂都可在本网站选购。 |