CAS NO: | 2095109-82-1 |
包装 | 价格(元) |
100mg | 电议 |
250mg | 电议 |
500mg | 电议 |
生物活性 | PAD2-IN-1, a benzimidazole-based derivative, is a potent and selectiveprotein arginine deiminase2 (PAD2)inhibitor. PAD2-IN-1 shows superior selectivity forPAD2over PAD4 (95-fold) and PAD3 (79-fold)[1]. |
IC50& Target | Protein Arginine Deiminase 2 (PAD2)[1] |
体外研究 (In Vitro) | In the target engagement assay, the EC50of PAD2-IN-1 (compound 32a) is 8.3 μM in HEK293T/PAD2 cells, the enhanced potency of PAD2-IN-1 overcomes its relatively poor ability to enter cells[1]. |
分子量 | 480.53 |
Formula | C25H29FN6O3 |
CAS 号 | 2095109-82-1 |
运输条件 | Room temperature in continental US; may vary elsewhere. |
储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |