| CAS NO: | 39552-01-7 |
| 包装: | 1mg |
| 市场价: | 2678元 |
| Cas No. | 39552-01-7 |
| 别名 | (±)-苯呋洛尔；氧茚心安 |
| Canonical SMILES | CC(C1=CC2=CC=CC(OCC(O)CNC(C)C)=C2O1)=O |
| 分子式 | C16H21NO4 |
| 分子量 | 291.34 |
| 溶解度 | Soluble in DMSO |
| 储存条件 | Store at -20°C |
| General tips | For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while. |
| Shipping Condition | Evaluation sample solution : ship with blue ice All other available size: ship with RT , or blue ice upon request |
| 产品描述 | (±)-Befunolol is a β-adrenoceptor blocking agent. A β-adrenoceptor blocking agent, Befunolol, is found to has intrinsic sympathomimetic activities in isolated right atria, trachea and taenia caecum of guinea pig (intrinsic activities are 0.22-0.28). The pD2-values of Befunolol estimated in the isolated organs are significantly different from its pA2-values against isoprenaline. Befunolol interacts with the beta-adrenoceptor where there may be two different sites: one site for agonistic action and the other for competitive antagonistic action. The intrinsic activity of Befunolol may be equal to its selectivity for both the sites[1]. [1]. Takayanagi I, et al. A beta-adrenoceptor blocking agent, befunolol as a partial agonist in isolated organs. Gen Pharmacol. 1985;16(3):265-7. |
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