CAS NO: | 1415560-64-3 |
包装 | 价格(元) |
5mg | 电议 |
10mg | 电议 |
50mg | 电议 |
CAS: | 1415560-64-3 |
分子式: | C29H27F3N4O7S |
分子量: | 632.61 |
纯度: | >98% |
溶解性: | DMSO |
存储: | Powder -20℃ 3 years; 4℃ 2 years In solvent -80℃ 6 months; -20℃ 1 month |
研究领域: | Inflammation/Immunology |
Target: | IC50: 3.2 pM (PDE4B)[1] |
描述: | GSK 256066 Trifluoroacetate is a selective PDE4B(equal affinity to isoforms A-D) inhibitor with IC50 of 3.2 pM, >380,000-fold selectivity versus PDE1/2/3/5/6 and >2500-fold selectivity against PDE4B versus PDE7. |