CAS NO: | 1936421-41-8 |
包装 | 价格(元) |
5mg | 电议 |
10mg | 电议 |
CAS: | 1936421-41-8 |
分子式: | C27H32F2N6O2 |
分子量: | 510.58 |
纯度: | >98% |
溶解性: | DMSO |
存储: | -20℃, stored under nitrogen. In solvent : -80℃, 6 months; -20℃, 1 month (stored under nitrogen) |
研究领域: | Cancer |
Target: | IC50: 1.1 nM (CBP), 12 nM (BRET), 4200 nM (BRD4(1)) |
描述: | GNE-049 is a highly potent and selective CBP inhibitor with an IC50 of 1.1 nM in TR-FRET assay. GNE-049 also inhibits BRET and BRD4(1) with IC50s of 12 nM and 4200 nM, respectively. |