CAS NO: | 1044870-39-4 |
包装 | 价格(元) |
10mg | 电议 |
50mg | 电议 |
100mg | 电议 |
产品名称: | 阿帕他隆 |
CAS: | 1044870-39-4 |
分子式: | C20H22N2O5 |
分子量: | 370.40 |
纯度: | >98% |
溶解性: | DMSO |
存储: | Powder -20℃ 3 years; 4℃ 2 years In solvent -80℃ 6 months;-20℃ 1 month |
研究领域: | Cancer |
Target: | IC50: 510±41 nM (BD2), 87±10 μM (BD1)[1] |
描述: | Apabetalone (RVX-208) is an inhibitor of BET transcriptional regulators with selectivity for the second bromodomain. The IC50s are 87±10 μM and 0.51±0.041 μM for BD1 and BD2, respectively. |