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Levetimide
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
Levetimide图片
CAS NO:21888-99-3
包装与价格:
包装价格(元)
10mM (in 1mL DMSO)电议
10mg电议
50mg电议
100mg电议
200mg电议

产品介绍
Levetimide 是一种有效的立体选择性 [3H](+)pentazocine 结合抑制剂,Ki 为 2.2 nM。
Cas No.21888-99-3
Canonical SMILESO=C(N1)[C@](C2=CC=CC=C2)(CCC1=O)C3CCN(CC3)CC4=CC=CC=C4
分子式C23H26N2O2
分子量362.46
溶解度DMSO: ≥ 100 mg/mL (275.89 mM)
储存条件Store at -20°C
General tipsFor obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.
Shipping ConditionEvaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request
产品描述

Levetimide is a potent and stereoselective inhibitor of [3H](+)pentazocine binding, with a Ki of 2.2 nM[1].

Levetimide potently inhibits [3H]DTG binding although without stereoselectivity (Ki value of 103 nM) [1].

[1]. DeHaven-Hudkins DL, et al. Binding of dexetimide and levetimide to [3H](+)pentazocine- and [3H]1,3-di(2-tolyl)guanidine-defined sigma recognition sites. Life Sci. 1991;49(18):PL135-9.