Cyclapolin 9 是一种有效的、选择性的和 ATP 竞争性的 polo 样激酶 1 (PLK1) 抑制剂,IC50 为 500 nM。 Cyclapolin 9 对其他激酶无活性。
Cas No. | 40533-25-3 |
化学名 | 2-carbamoyl-7-nitro-5-(trifluoromethyl)benzo[d]thiazole 3-oxide |
Canonical SMILES | FC(F)(F)C1=CC(N(=C2C(N)=O)=O)=C(S2)C(N(=O)=O)=C1 |
分子式 | C9H4F3N3O4S |
分子量 | 307.21 |
溶解度 | <7.68mg/ml in DMSO |
储存条件 | Store at -20℃ |
General tips | For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while. |
Shipping Condition | Evaluation sample solution : ship with blue ice All other available size: ship with RT , or blue ice upon request |