| CAS NO: | 1185160-65-9 |
| 包装 | 价格(元) |
| 500 μg | 电议 |
| 1mg | 电议 |
| Cas No. | 1185160-65-9 |
| 别名 | 盐酸托哌酮 d10 (盐酸盐) |
| Canonical SMILES | CC1=CC=C(C(C(CN2C([2H])([2H])C([2H])([2H])C([2H])([2H])C([2H])([2H])C2([2H])[2H])C)=O)C=C1.Cl |
| 分子式 | C16H13D10NO.HCl |
| 分子量 | 291.9 |
| 储存条件 | Store at 2°C to 8°C |
| General tips | For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while. |
| Shipping Condition | Evaluation sample solution : ship with blue ice All other available size: ship with RT , or blue ice upon request |
| 产品描述 | Tolperisone-d10is intended for use as an internal standard for the quantification of tolperisone by GC- or LC-MS. Tolperisone is a piperidine that acts as an inhibitor of voltage-gated sodium channels with an IC50value of 198 µM, for inhibition of peak sodium currents evoked by step depolarizations in dorsal root ganglion (DRG) neurons,in vitro.1Tolperisone acts as an antispastic agent that attenuates monosynaptic, disynaptic, and polysynaptic reflux response to dorsal root stimulationin vivo. Formulations containing tolperisone are used as analgesics and muscle relaxants. 1.Kocsis, P., Farkas, S., Fodor, L., et al.Tolperisone-type drugs inhibit spinal reflexes via blockade of voltage-gated sodium and calcium channelsJ. Pharmacol. Exp. Ther.315(3)1237-1246(2005) |
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