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EHMT2-IN-1
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
EHMT2-IN-1图片
CAS NO:2230849-55-3
包装与价格:
包装价格(元)
10mM (in 1mL DMSO)电议
5mg电议
10mg电议
25mg电议

产品介绍
EHMT2-IN-1是一种有效的EHMT抑制剂,对EHMT1多肽,EHMT2多肽和细胞内EHMT2的IC50均小于100nM。用于血液疾病或癌症的研究。
Cas No.2230849-55-3
Canonical SMILESCOC1=C(N2N=CC(CNC)=C2)C=C(NC3=NC(NC)=CC(C)=N3)C=C1
分子式C18H23N7O
分子量353.42
溶解度DMSO : 55 mg/mL (155.62 mM)
储存条件Store at -20°C
General tipsFor obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.
Shipping ConditionEvaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request
产品描述

EHMT2-IN-1 is a potent EHMT inhibitor, with IC50s of all<100 nM for EHMT1 peptide, EHMT2 peptide and cellular EHMT2. Used in the research of blood disorder or cancer[1]. EHMTI PEP|<100 nM (IC50)|EHMT2 PEP|<100 nM (IC50)|EHMT2 ICW|<100 nM (IC50)

EHMT2-IN-1 (Compound 108) potent EHMT inhibitor, with IC50s of all<100 nM for EHMT1 peptide, EHMT2 peptide and cellular EHMT2[1].

[1]. John Emmerson Campbell, et al. Amine-substituted heterocyclic compounds as ehmt2 inhibitors and methods of use thereof. WO2018118842A1