CAS NO: | 2230849-55-3 |
包装 | 价格(元) |
10mM (in 1mL DMSO) | 电议 |
5mg | 电议 |
10mg | 电议 |
25mg | 电议 |
Cas No. | 2230849-55-3 |
Canonical SMILES | COC1=C(N2N=CC(CNC)=C2)C=C(NC3=NC(NC)=CC(C)=N3)C=C1 |
分子式 | C18H23N7O |
分子量 | 353.42 |
溶解度 | DMSO : 55 mg/mL (155.62 mM) |
储存条件 | Store at -20°C |
General tips | For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while. |
Shipping Condition | Evaluation sample solution : ship with blue ice All other available size: ship with RT , or blue ice upon request |
产品描述 | EHMT2-IN-1 is a potent EHMT inhibitor, with IC50s of all<100 nM for EHMT1 peptide, EHMT2 peptide and cellular EHMT2. Used in the research of blood disorder or cancer[1]. EHMTI PEP|<100 nM (IC50)|EHMT2 PEP|<100 nM (IC50)|EHMT2 ICW|<100 nM (IC50) EHMT2-IN-1 (Compound 108) potent EHMT inhibitor, with IC50s of all<100 nM for EHMT1 peptide, EHMT2 peptide and cellular EHMT2[1]. [1]. John Emmerson Campbell, et al. Amine-substituted heterocyclic compounds as ehmt2 inhibitors and methods of use thereof. WO2018118842A1 |