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Ostarine
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
Ostarine图片
CAS NO:841205-47-8
包装与价格:
包装价格(元)
5mg电议
10mg电议
50mg电议
100mg电议
200mg电议
500mg电议

产品介绍
Ostarine(MK-2866; GTX-024)是选择性雄激素受体调节剂,ED50为0.44 mg/day。
Cas No.841205-47-8
Canonical SMILESFC(F)(C1=CC(NC([C@](C)(COC2=CC=C(C=C2)C#N)O)=O)=CC=C1C#N)F
分子式C19H14F3N3O3
分子量389.33
溶解度DMSO: ≥ 100 mg/mL (256.85 mM); Water:< 0.1 mg/mL (insoluble)
储存条件Store at -20°C
General tipsFor obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.
Shipping ConditionEvaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request
产品描述

Ostarine(MK-2866; GTX-024) is a modulator of human androgen receptor.IC50 value:Target: androgen receptorOstarine (MK-2866) is an androgen receptor modulator (SARM) with an ED50 of 0.44 mg/day. Ostarine (MK-2866) has anabolic activity. Lack of PSA increases in men and hair growth in women further corroborated selective anabolic effects of Ostarine (MK-2866). Ostarine (MK-2866) also resulted in a dose-dependent decrease in LDL and HDL cholesterol levels, with the average LDL/HDL ratio for all doses remaining in the low cardiovascular risk catergory.

[1]. Thevis M, et al. Trafficking of drug candidates relevant for sports drug testing: detection of non-approved therapeutics categorized as anabolic and gene doping agents in products distributed via the Internet.Drug Test Anal. 2011 May;3(5):331-6. doi: 10.1002/dta.283. [2]. Zilbermint MF, et al. Nonsteroidal selective androgen receptor modulator Ostarine in cancer cachexia. Nonsteroidal selective androgen receptor modulator Ostarine in cancer cachexia.