| CAS NO: | 1308833-36-4 |
| 包装 | 价格(元) |
| 1mg | 电议 |
| 5mg | 电议 |
| 10mg | 电议 |
| 25mg | 电议 |
| Cas No. | 1308833-36-4 |
| 别名 | (9H-芴-9-基)甲基((S)-1(((S)-6-(叔丁氧基羰基)氨基-1-((4-甲基-2-氧代-1,2-二氢喹啉-7-基)氨基)-1-氧代己-2-基)氨基)-3-环己基-1-氧代丙-2-基)氨基甲酸叔丁酯 |
| Canonical SMILES | CC(C1=CC=C(C=C1N2)NC([C@H](CCCCNC(OC(C)(C)C)=O)NC([C@H](CC3CCCCC3)NC(OCC4C5=CC=CC=C5C6=CC=CC=C64)=O)=O)=O)=CC2=O |
| 分子式 | C45H55N5O7 |
| 分子量 | 778 |
| 储存条件 | -20°C |
| General tips | For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while. |
| Shipping Condition | Evaluation sample solution : ship with blue ice All other available size: ship with RT , or blue ice upon request |
| 产品描述 | CYM 2503 is a positive allosteric modulator (PAM) of the galanin-2 (GAL2) receptor.1It enhances the production of inositol monophosphate (IP1) induced by galanin in HEK293 cells expressing the GAL2receptor (EC50= 0.69 µM). CYM 2503 (60 mg/kg) increases the latency to first electrographic and behavioral seizures and reduces mortality in a lithium-pilocarpine (Li-pilocarpine) rat model of status epilepticus. 1.Lu, X., Roberts, E., Xia, F., et al.GalR2-positive allosteric modulator exhibits anticonvulsant effects in animal modelsProc. Natl. Acad. Sci. USA107(34)15229-15234(2010) |
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