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BZAD-01
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
BZAD-01图片
CAS NO:305339-41-7
包装与价格:
包装价格(元)
5mg电议
10mg电议
25mg电议
50mg电议

产品介绍
BZAD-01 是一种有效的,选择性和具有口服活性的 NMDA NR2B 抑制剂,Ki 值为 72 nM。BZAD-01 可以改善姿势不对称以及阿扑吗啡引起的旋转。
Cas No.305339-41-7
分子式C16H12F6N2O
分子量362.27
溶解度Methanol : 250 mg/mL (690.09 mM; Need ultrasonic)|DMSO : 100 mg/mL (276.04 mM; Need ultrasonic)
储存条件4°C, protect from light
General tipsFor obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.
Shipping ConditionEvaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request
产品描述

BZAD-01 is a potent, selective and orally active inhibitor of NMDA NR2B subunit, with a Ki of 72 nM. BZAD-01 can improve postural asymmetry as well as Apomorphine-induced rotation[1].

[1]. Truong L, et, al. Behavioural effects of a selective NMDA NR1A/2B receptor antagonist in rats with unilateral 6-OHDA+parafascicular lesions. Brain Res Bull. 2009 Feb 16;78(2-3):91-6.