您好,欢迎来到试剂仪器网! [登录] [免费注册]
试剂仪器网
位置:首页 > 产品库 > Inupadenant
立即咨询
咨询类型:
     
*姓名:
*电话:
*单位:
Email:
*留言内容:
请详细说明您的需求。
*验证码:
 
Inupadenant
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
Inupadenant图片
CAS NO:2246607-08-7
包装与价格:
包装价格(元)
1mg电议
5mg电议

产品介绍
Inupadenant (EOS-850) 是一种具有口服活性的,高选择性 A2A 受体拮抗剂。Inupadenant 不能透过血脑屏障。Inupadenant 具有抗肿瘤活性。
Cas No.2246607-08-7
别名EOS-850
分子式C25H26F2N8O4S2
分子量604.65
General tipsFor obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.
Shipping ConditionEvaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request
产品描述

Inupadenant is an orally active, highly selective A2A receptor antagonist. Inupadenant is not brain-penetrant. Inupadenant has potent anti-tumor activity[1].

[1]. Laurence Buisseret, et al. Phase 1 trial of the adenosine A2Areceptor antagonist inupadenant (EOS-850): Update on tolerability, and antitumor activity potentially associated with the expression of the A2A receptor within the tumor. Journal of Clinical Oncology. Volume 39, Issue 15_suppl.