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NSC 694621
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
NSC 694621图片
CAS NO:104857-29-6
包装与价格:
包装价格(元)
10mg电议
25mg电议
50mg电议
100mg电议

产品介绍
NSC 694621 是一种有效的 PCAF 抑制剂,其 IC50 值为 5.71 µM (PCAF/H31-21)。NSC 694621 具有较好的抗癌活性,能抑制癌细胞的增殖。
Cas No.104857-29-6
分子式C13H10N2O2S
分子量258.3
储存条件Store at -20°C
General tipsFor obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.
Shipping ConditionEvaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request
产品描述

IC50: 5.71 µM (PCAF/H31-21)[1].

NSC 694621 is a potentPCAFinhibitor, with anIC50of 5.71 µM (PCAF/H31-21). NSC 694621 exhibits good activity of inhibiting the proliferation of cancer cells[1].

NSC 694621 (25 µM; 72 h) exhibits antiproliferative effect to SK-N-SH and HCT116 cells[1].

Cell Proliferation Assay[1]

Cell Line:SK-N-SH, HCT116 cells
Concentration:25 µM
Incubation Time:72 h
Result:Showed antiproliferative effect to SK-N-SH and HCT116 cells with GI50of 19.2 µM and growth inhibition of 29%, respectively.