CGP 13501 is a positive allosteric modulator of GABAB receptor. In cells expressing GABAB(1b+2) receptors, CGP13501 increased GTPγ[35S] binding at Gαi1/3. References: Mannoury la Cour C, Herbelles C, Pasteau V, de Nanteuil G, Millan MJ. Influence of positive allosteric modulators on GABA(B) receptor coupling in rat brain: a scintillation proximity assay characterisation of G protein subtypes. J Neurochem. 2008 Apr;105(2):308-23. PubMed PMID: 18021295.

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CAS：56189-68-5