CGP 46381 is a brain penetrant, selective GABAB receptor antagonist (IC50 = 4.9 μM). References: Ishige K, Endo H, Saito H, Ito Y. Repeated administration of CGP 46381, a gamma-aminobutyric acidB antagonist, and ethosuximide suppresses seizure-associated cyclic adenosine 3'5' monophosphate response element- and activator protein-1 DNA-binding activities in lethargic (lh/lh) mice. Neurosci Lett. 2001 Jan 19;297(3):207-10. PubMed PMID: 11137764.

纯度：≥98%

CAS：123691-14-5