DCG066 is a G9a inhibitor. DCG066 can bind directly to G9a and inhibit methyltransferase activity in vitro. It exhibits low cytotoxicity in leukemia cell lines with high levels of G9a expression, including K562. References: Kondengaden SM, Luo LF, Huang K, Zhu M, Zang L, Bataba E, Wang R, Luo C, Wang B, Li KK, Wang PG. Discovery of novel small molecule inhibitors of lysine methyltransferase G9a and their mechanism in leukemia cell lines. Eur J Med Chem. 2016 Oct 21;122:382-393. doi: 10.1016/j.ejmech.2016.06.028. Epub 2016 Jun 21. PubMed PMID: 27393948.

纯度：≥98%

CAS：494786-13-9