Burapitant, formerly known as SSR 240600, is a potent and selective NK1 receptor antagonist. SSR240600 is found to effectively antagonize various NK1 receptor-mediated as well as stress-mediated effects in the guinea pig. References: PA(C)rez S, Tierney A, Deniau JM, Kemel ML. Tachykinin regulation of cholinergic transmission in the limbic/prefrontal territory of the rat dorsal striatum: implication of new neurokinine 1-sensitive receptor binding site and interaction with enkephalin/mu opioid receptor transmission. J Neurochem. 2007 Dec;103(6):2153-63. Epub 2007 Oct 18. PubMed PMID: 17949415.

纯度：≥98%

CAS：537034-22-3