Epelsiban besylate is an orally bioavailable drug which acts as a selective, sub-nanomolar (Ki=0.13 nM) oxytocin receptor antagonist with >31000-fold selectivity over the related vasopressin receptors. It is being developed by GlaxoSmithKline for the treatment of premature ejaculation in men. References: Mahar KM, Stier B, Fries M, McCallum SW. A single- and multiple-dose study to investigate the pharmacokinetics of epelsiban and its metabolite, GSK2395448, in healthy female volunteers. Clin Pharmacol Drug Dev. 2015 Nov;4(6):418-26. doi: 10.1002/cpdd.210. Epub 2015 Aug 26. PubMed PMID: 27137713.

纯度：≥98%

CAS：1159097-48-9