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FK-888
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
CAS NO:138449-07-7
包装:50mg, 100mg, 250mg
规格:≥98%

产品介绍

FK-888 is a selective, high affinity tachykinin NK1 receptor antagonist (Ki = 0.69 nM) that exhibits 320-fold selectivity for human over rat NK1 receptors. FK-888 inhibits substance P-induced contraction of isolated guinea pig trachea (IC50 = 32 nM) and inhibits substance P-induced airway constriction in vivo. References: Esposito V, Linard C, Wysocki J, Griffiths NM, Mathe D. A substance P receptor antagonist (FK 888) modifies gut alterations induced by ionizing radiation. Int J Radiat Biol. 1998 Nov;74(5):625-32. PubMed PMID: 9848281.

纯度:≥98%

CAS:138449-07-7