Setin-1 is the most potent inhibitor of Set7 that acts by inhibiting the KMTase G9a. References: Kashyap S, Sandler J, Peters U, Martinez EJ, Kapoor TM. Using 'biased-privileged' scaffolds to identify lysine methyltransferase inhibitors. Bioorg Med Chem. 2014 Apr 1;22(7):2253-60. doi: 10.1016/j.bmc.2014.02.024. Epub 2014 Feb 28. PubMed PMID: 24650704; PubMed Central PMCID: PMC4038709.

纯度：≥98%

CAS：1313802-67-3