SB258585 Hydrochloride is a potent, selective antagonist of the serotonin 5-HT6 receptor (pKi = 8.53). It exhibits over 100-fold selectivity for 5-HT6 over other 5-HT, dopamine, and α-adrenergic receptors. References: Yun HM, Rhim H. 5-HT6 receptor ligands, EMD386088 and SB258585, differentially regulate 5-HT6 receptor-independent events. Toxicol In Vitro. 2011 Dec;25(8):2035-40. doi: 10.1016/j.tiv.2011.08.004. Epub 2011 Aug 16. PubMed PMID: 21864673.

纯度：≥98%

CAS：1216468-02-8