RX821002 is a potent, selective α2-adrenoceptor antagonist with very low affinity for imidazoline sites. RX821002 exhibits selectivity for the α2D over the α2A subtypes (pKd values are 9.7 and 8.2 respectively). References: Sandner G, Angst MJ, Guiberteau T, Guignard B, Nehlig A. Effects of caffeine or RX821002 in rats with a neonatal ventral hippocampal lesion. Front Behav Neurosci. 2014 Jan 28;8:15. doi: 10.3389/fnbeh.2014.00015. eCollection 2014. PubMed PMID: 24478661; PubMed Central PMCID: PMC3904090.

纯度：≥98%

CAS：102575-24-6