ATSP-7041 is a potent and selective dual inhibitor of mdm2 (ki = 0.9 nm) and mdmx (ki = 7 nm) References: Partridge AW, Kaan HYK, Juang YC, Sadruddin A, Lim S, Brown CJ, Ng S, Thean D, Ferrer F, Johannes C, Yuen TY, Kannan S, Aronica P, Tan YS, Pradhan MR, Verma CS, Hochman J, Chen S, Wan H, Ha S, Sherborne B, Lane DP, Sawyer TK. Incorporation of Putative Helix-Breaking Amino Acids in the Design of Novel Stapled Peptides: Exploring Biophysical and Cellular Permeability Properties. Molecules. 2019 Jun 20;24(12). pii: E2292. doi: 10.3390/molecules24122292. PubMed PMID: 31226791.

纯度：≥98%

CAS：1451197-99-1