Tecastemizole (Norastemizole)，Astemizole 的主要代谢物，是一种有效的、选择性的 H1 receptor 拮抗剂。Tecastemizole 具有抗炎活性。
货号:ajcx37822
CAS:75970-99-9
分子式:C19H21FN4
分子量：324.4
溶解度:DMSO : 100 mg/mL (308.26 mM; ultrasonic and warming and heat to 60°C)
纯度：98%
存储：Store at -20°C
库存：现货

Background:

Tecastemizole (Norastemizole), a major metabolite of Astemizole, is a potent and selective H1 receptor antagonist. Tecastemizole shows anti-inflammatory activities[1].

[1]. Lever R, et al. Effect of tecastemizole on pulmonary and cutaneous allergic inflammatory responses. Clin Exp Allergy. 2007 Jun;37(6):909-17.