规格: | 98% |
分子量: | 367.9 |
包装 | 价格(元) |
500ug | 电议 |
1mg | 电议 |
Background:
5-hydroxy Saxagliptin is a major active metabolite of saxagliptin . 5-hydroxy Saxagliptin inhibits dipeptidyl peptidase 4 (DPP-4; Ki = 2.6 nM for human recombinant enzyme). It is selective for DPP-4 over DPP-8 and DPP-9 (Kis = 2,495 and 423 nM, respectively, for human recombinant enzymes).