CAS NO: | 84449-90-1 |
规格: | ≥98% |
包装 | 价格(元) |
1g | 电议 |
2g | 电议 |
5g | 电议 |
10g | 电议 |
Description: Raloxifene (also known as LY156758; LY-139481) is a selective estrogen antagonist or estrogen strogen receptor modulator (SERM), which inhibits human cytosolic aldehyde oxidase-catalyzed phthalazine oxidation activity with IC50 of 5.7 nM. Raloxifene belongs to the benzothiophene class of estrogen strogen receptor modulator (SERM). Raloxifene binds to estrogen receptors as a mixed estrogen agonist/antagonist; it displays both an ER-α-selective partial agonist/antagonist effect and a pure ER-ss-selective antagonist effect. References: Drug Metab Dispos. 2004 Jan;32(1):89-97; Endocrinology. 1996 May;137(5):2075-84. Related CAS #: 84449-90-1 (free base) 82640-04-8 or 84449-90-1 (HCl)
纯度:≥98%
CAS:84449-90-1