规格: | 98% |
分子量: | 496.03 |
包装 | 价格(元) |
5mg | 电议 |
25mg | 电议 |
Background:
Potent ghrelin receptor inverse agonist (IC50 = 4.6 nM). Orally bioavailable and exhibits reasonable brain penetration.
Kung et al (2012) Identification of spirocyclic piperidine-azetidine inverse agonists of the ghrelin receptor. Bioorg.Med.Chem.Lett. 22 5410 PMID:22677316