规格: | 98% |
分子量: | 428.31 |
包装 | 价格(元) |
1mg | 电议 |
5mg | 电议 |
10mg | 电议 |
25mg | 电议 |
Background:
(R)-MLN-4760, the R-enantiomer of MLN-4760, is an ACE2 inhibitor, with an IC50 of 8.4 µM. (R)-MLN-4760 is the less active isomer[1].
(R)-MLN-4760 (compound 16RS) is the less active isomer of MLN-4760[1].
参考文献:
[1]. Dales NA, et, al. Substrate-based design of the first class of angiotensin-converting enzyme-related carboxypeptidase (ACE2) inhibitors. J Am Chem Soc. 2002 Oct 9;124(40):11852-3.