Radequinil (AC-3933) 是一种苯二氮卓类受体 (BzR) 部分反向激动剂。AC-3933 与 GABA(-) 和 GABA(+) 配体结合，Ki 分别为 5.15 和 6.11 nM。
货号:ajcx39726
CAS:219846-31-8
分子式:C18H14N4O3
分子量：334.33
溶解度:DMSO : 10 mg/mL (29.91 mM; ultrasonic and warming and heat to 60°C)
纯度：98%
存储：Store at -20°C
库存：现货

Background:

Radequinil (AC-3933) is a benzodiazepine receptor (BzR) partial inverse agonist. AC-3933 binds to GABA(-) and GABA(+) ligand with Kis of 5.15 and 6.11 nM, respectively[1].

[1]. Hashimoto T, et al. Pharmacological properties of AC-3933, a novel benzodiazepine receptor partial inverse agonist. Neuroscience. 2014 Jan 3;256:352-9.