C21H23D11O2
货号:ajcx24532
CAS:N/A
分子式:C21H23D11O2
分子量：329.6
溶解度:DMF: 10 mg/ml,DMSO: 15 mg/ml,Ethanol: 10 mg/ml,Methanol: 12.5 mg/ml
纯度：98%
存储：Store at -20°C
库存：现货

Background:

(±)-CP 47,497-d₁₁(exempt preparation) contains eleven deuterium atoms at the 4, 4', 5, 5', 6, 6', 7, 7', 8, 8, and 8 positions. It is intended for use as an internal standard for the quantification of (±)-CP 47,497 (exempt preparation) by GC-or LC-mass spectrometry. CP 47,497 is a monophenol cannabimimetic compound that binds the central cannabinoid (CB₁) receptor with a K_ivalue of 2.2 nM.^1,2It is equivalent in analgesic potency to δ⁹-THC and exhibits other CB biological activities as well.

1.Huffman, J.W., Thompson, A.L.S., Wiley, J.L., et al.Synthesis and pharmacology of 1-deoxy analogs of CP-47,497 and CP-55,940Bioorganic & Medicinal Chemistry16322-335(2008) 2.Melvin, L.S., Milne, G.M., Johnson, M.R., et al.Structure-activity relationships for cannabinoid receptor-binding and analgesic activity: Studies of bicyclic cannabinoid analogsMol. Pharmacol.44(5)1008-1015(1993)