Subtype-selective agonist of α4β2 nicotinic receptors,orally active
CAS：375815-87-5
分子式：C13H13N3.C4H6O6
分子量：361.35
纯度：98%
存储：Store at -20°C

Background:

Varenicline Tartrate(CP 526555;Champix) is a nicotinic receptor partial agonist; it stimulates nicotine receptors more weakly than nicotine itself does.IC50 value:Target: α4β2 nAChRVarenicline(CP 526555; Champix; Chantix) is a prescription medication used to treat smoking addiction. As a partial agonist it both reduces cravings for and decreases the pleasurable effects of cigarettes and other tobacco products. Through these mechanisms Varenicline(CP 526555; Champix; Chantix) can assist some patients to quit smoking.

参考文献:
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[5]. Varenicline