Raloxifene 6-glucuronide is a metabolite of the selective estrogen receptor modulator raloxifene.
CAS：174264-50-7
分子式：C34H35NO10S
分子量：649.7
纯度：98%
存储：Store at -20°C

Background:

Raloxifene 6-glucuronide is a metabolite of the selective estrogen receptor modulator raloxifene . It is formed from raloxifene via the UDP-glucuronosyltransferase (UGT) isoforms UGT1A1 and UGT1A8. It binds to the estrogen receptor with an IC50 value of 290 nM. Unlike raloxifene, raloxifene 6-glucuronide does not inhibit the voltage-gated potassium channel Kv4.3.